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A multi-centre, open label phase 2 trial investigating the effect of evolocumab in addition to chemotherapy or androgen receptor signalling inhibitor therapy on the circulating lipid profile of men with metastatic castration-resistant prostate cancer

ACTRN 12622001003763

Brief Summary

Elevated lipids called ceramides are associated with poorer outcomes in men with prostate cancer. Statins, a class of drug that reduces lipid levels, have been shown to be somewhat helpful in reversing this poor prognostic lipid signature, however only in a subset of men with metastatic castration-resistant prostate cancer (mCRPC) (i.e. those that are resistant to anti-androgen treatment). Therefore, other more potent or targeted lipid lowering drugs such as the anti-proprotein convertase subtilisin/kexin type 9 (PCSK9) monoclonal antibody (PCSK9) inhibitor evolocumab may be required. This study aims to assess whether evolocumab reduces ceramide levels in men with mCRPC commencing chemotherapy or androgen receptor signaling inhibitors (ARSI) therapy.

Intervention/Treatment

  • Drug: Evolocumab.
  • Chemotherapy.
  • Androgen receptor signaling inhibitor (ARSI) therapy.
  • Poly ADP ribose polymerase inhibitor (PARPI) therapy.
  • Lutetium-177 prostatespecific membrane antigen (PSMA) therapy.

Inclusion Criteria:

  1. Males with mCRPC (as per prostate cancer working group (PCWG3)) AND commencing docetaxel, cabazitaxel, abiraterone or enzalutamide, olaparib or lutetium for disease progression.
  2. Age > 18 yrs.
  3. WHO ECOG performance status 0-2.
  4. Histological confirmation of prostate cancer.
  5. Adequate hepatic function with serum total bilirubin > 1.5 x upper limit of normal (ULN) range and ALT and AST > 2.5x upper limit of normal range (or < 5.0 times ULN with documented liver metastases), serum albumin > 25 g/L, and ALP > 5x upper limit of normal range.
  6. Adequate renal function (with calculated creatinine clearance >50 ml/min based on the Cockcroft-Gault method, 24 hour urine or GFR scan) and serum creatinine > 1.5 x upper limit of normal range.
  7. Demonstrated positivity for high-risk circulating plasma lipid profile on Liquid chromatography–mass spectrometry (LCMS).
  8. Willing and able to comply with all study requirements, including treatment and biospecimen collection.
  9. Signed written informed consent.

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